Browsing publications by Professor Jane Endicott

Newcastle AuthorsTitleYear
Dr Alison Hole
Dr Sonja Baumli
Professor Jane Endicott
Professor Martin Noble
Comparative Structural and Functional Studies of 4-(Thiazol-5-yl)-2-(phenylamino)pyrimidine-5-carbonitrile CDK9 Inhibitors Suggest the Basis for Isotype Selectivity2013
Professor Martin Noble
Professor Jane Endicott
Substituted 4-(Thiazol-5-yl)-2-(phenylamino)pyrimidines Are Highly Active CDK9 Inhibitors: Synthesis, X-ray Crystal Structures, Structure-Activity Relationship, and Anticancer Activities2013
Professor Martin Noble
Professor Jane Endicott
Structural and functional characterization of Rpn12 identifies residues required for Rpn10 proteasome incorporation2012
Professor Jane Endicott
Synthesis and in Vitro Evaluation of Selective CDK9 Inhibitors2012
Dr Sonja Baumli
Dr Alison Hole
Professor Martin Noble
Professor Jane Endicott
The CDK9 C-helix Exhibits Conformational Plasticity That May Explain the Selectivity of CAN5082012
Dr Sonja Baumli
Dr Alison Hole
Lan-zhen Wang
Professor Martin Noble
Professor Jane Endicott
et al.		The CDK9 Tail Determines the Reaction Pathway of Positive Transcription Elongation Factor b2012
Professor Jane Endicott
Professor Martin Noble
The Structural Basis for Control of Eukaryotic Protein Kinases2012
Professor Jane Endicott
The ubiquitin-associated (UBA) 1 domain of Schizosaccharomyces pombe Rhp23 is essential for the recognition of ubiquitin-proteasome system substrates both in Vitro and in Vivo2012
Dr Ian Hardcastle
Alex Liu
Dr Eric Valeur
Anna Watson
Shafiq Ahmed
et al.		Isoindolinone Inhibitors of the Murine Double Minute 2 (MDM2)-p53 Protein-Protein Interaction: Structure-ActivityStudies Leading to Improved Potency2011
Dr Karim Bennaceur
Dr Catherine Drummond
Professor Jane Endicott
Professor Bernard Golding
Professor Roger Griffin
et al.		MDM2-p53 protein-protein interaction inhibitors: A-ring substituted isoindolinones2011
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